GPR87
This gene encodes a G protein-coupled receptor and is located in a cluster of G protein-couple receptor genes on chromosome 3. The encoded protein has been shown to be overexpressed in lung squamous cell carcinoma (PMID:18057535) and regulated by p53.
Full Name
G protein-coupled receptor 87
Function
Receptor for lysophosphatidic acid (LPA). Necessary for p53/TP53-dependent survival in response to DNA damage.
Biological Process
G protein-coupled receptor signaling pathway Source: GO_Central
Negative regulation of adenylate cyclase activity Source: InterPro
Negative regulation of adenylate cyclase activity Source: InterPro
Cellular Location
Cell membrane
Topology
Extracellular: 1-47
Helical: 48-68
Cytoplasmic: 69-75
Helical: 76-96
Extracellular: 97-116
Helical: 117-137
Cytoplasmic: 138-159
Helical: 160-180
Extracellular: 181-208
Helical: 209-229
Cytoplasmic: 230-256
Helical: 257-277
Extracellular: 278-297
Helical: 298-318
Cytoplasmic: 319-358
Helical: 48-68
Cytoplasmic: 69-75
Helical: 76-96
Extracellular: 97-116
Helical: 117-137
Cytoplasmic: 138-159
Helical: 160-180
Extracellular: 181-208
Helical: 209-229
Cytoplasmic: 230-256
Helical: 257-277
Extracellular: 278-297
Helical: 298-318
Cytoplasmic: 319-358
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Anti-GPR87 antibodies
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Target: GPR87
Host: Human
Antibody Isotype: IgG1
Specificity: Human
Clone: CBLG1-1647
Application*: F
Target: GPR87
Host: Mouse
Antibody Isotype: IgG2a, κ
Specificity: Human
Clone: EG1410
Application*: E
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For Research Use Only. Not For Clinical Use.
(P): Predicted
* Abbreviations
- AActivation
- AGAgonist
- APApoptosis
- BBlocking
- BABioassay
- BIBioimaging
- CImmunohistochemistry-Frozen Sections
- CIChromatin Immunoprecipitation
- CTCytotoxicity
- CSCostimulation
- DDepletion
- DBDot Blot
- EELISA
- ECELISA(Cap)
- EDELISA(Det)
- ESELISpot
- EMElectron Microscopy
- FFlow Cytometry
- FNFunction Assay
- GSGel Supershift
- IInhibition
- IAEnzyme Immunoassay
- ICImmunocytochemistry
- IDImmunodiffusion
- IEImmunoelectrophoresis
- IFImmunofluorescence
- IGImmunochromatography
- IHImmunohistochemistry
- IMImmunomicroscopy
- IOImmunoassay
- IPImmunoprecipitation
- ISIntracellular Staining for Flow Cytometry
- LALuminex Assay
- LFLateral Flow Immunoassay
- MMicroarray
- MCMass Cytometry/CyTOF
- MDMeDIP
- MSElectrophoretic Mobility Shift Assay
- NNeutralization
- PImmunohistologyp-Paraffin Sections
- PAPeptide Array
- PEPeptide ELISA
- PLProximity Ligation Assay
- RRadioimmunoassay
- SStimulation
- SESandwich ELISA
- SHIn situ hybridization
- TCTissue Culture
- WBWestern Blot
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